Expiration date: 01/2026
Release Form: pills.
Composition
1 tablet contains caffeine (as sodium benzoate) 0.1 g
Packaging: 6 pcs.
Pharmachologic effect
Analeptic, psychostimulant, cardiotonic. It has a stimulating effect on the central nervous system, increases the reflex excitability of the spinal cord, stimulates the respiratory and vasomotor centers, regulates and strengthens the processes of excitation in the cerebral cortex. It improves mental and physical performance, reduce fatigue and sleepiness. Increases force and heart rate (especially in high doses), increases blood pressure hypotension (not alter normal). Dilates blood vessels in skeletal muscle, heart, kidney, bronchus, narrows - abdominal organs. Improves the secretory activity of the stomach. It decreases platelet aggregation. It has a mild diuretic effect. Does central and peripheral adenosine receptors. It stabilizes the transmission of dopamine in synapses, beta-adrenergic synapses hypothalamus and the medulla oblongata, the cholinergic synapses of the cortex and the medulla oblongata, noradrenergic synapses. Effect of the drug largely depends on the nervous system of the patient, dosage of caffeine should therefore take into account the individual characteristics of neural activity.
Testimony
Diseases accompanied by inhibition of the central nervous system, cardiovascular system, respiratory system (drug poisoning, infectious diseases, etc.). When spasm of cerebral vessels, to improve mental and physical performance, to eliminate sleepiness, respiratory disorders, enuresis in children.
Contraindications
Severe hypertension, organic diseases of the cardiovascular system (including atherosclerosis), increased excitability, glaucoma, sleep disturbances, senile vozrast.Pobochnoe action
Anxiety, agitation, insomnia, tachycardia, arrhythmias, increased blood pressure, nausea, vomiting. Prolonged use may faint addictive (reduction of caffeine is associated with the formation of new cells in the brain adenosine receptors). Sudden discontinuation of caffeine can lead to increased inhibition of the CNS with symptoms of fatigue, lethargy and depression.
Dosing and Administration
The tablets are taken orally - on 0,025-0,1 g 2-3 times a day.
The maximum single dose for adults - 0.4 grams daily - 1 Year
Drug interactions
It reduces the effect of hypnotics, and narcotics, increases (improving bioavailability) - acetylsalicylic acid, paracetamol and other non-narcotic analgesics.. Improves absorption of ergotamine in the digestive tract.
Overdose
When abuse of caffeine (more than 300 mg per day, ie four cups of organic coffee, 150 ml) can cause anxiety, restlessness, tremor, headache, confusion, cardiac arrhythmia. In newborns (including premature) at a concentration in the blood plasma of 50 mg / ml may be toxic effects: anxiety, tachypnea, tachycardia, tremor, increased reflex Moro, at higher concentrations - cramps.
